Product name |
Flupirtine Maleate |
Appearance |
white solid |
Purity |
99%min |
CAS No. |
75507-68-5 |
EINECS No. |
278-225-0 |
MF. |
C19H21FN4O6 |
Grade Standard |
Medicine Grade |
Flupirtine maleate is a selective neuronal potassium channel openers, readily absorbed orally with analgesic, muscle relaxation and neuroprotective three efficacy, pain showed analgesic effects to a variety of causes. As in the hot plate test, intensity of flupirtine (ED50 32mg/Kg, Ig) is about half of the 2 times of paracetamol 10 times stronger. In the pulp electrical stimulation test of conscious dogs, the intensity of pain (ED50, 3.5mg/Kg, intragastric administration) was comparable to that of Zosin.
Flupirtine maleate is used as an analgesic for acute and chronic pain,in moderate-to-severe cases,Flupirtine maleate is also used for migraines.Flupirtine maleate has been noted for its neuroprotective properties,and Flupirtine maleate is being investigated for possible use in Creutzfeldt-Jakob disease,Alzheimer's disease,and multiple sclerosis.Flupirtine maleate has also been proposed as a possible treatment for Batten disease.
In the field of medicine use for the treatment of degenerative joint disease, neurological and cancer pain,migraine, headache and dysmenorrhea.